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Biochemistry

Statins

A class of drugs that lower LDL cholesterol by 30–55% — the cornerstone of heart-attack and stroke prevention.

Statins — a tablet blocking an enzyme, an artery clearing of plaque

Statins are the most prescribed drugs for lowering cholesterol. They block the liver enzyme HMG-CoA reductase — the key enzyme in cholesterol synthesis — which makes the liver take up "bad" LDL from the blood more actively.

By lowering LDL, statins slow the growth of atherosclerotic plaques and reliably reduce the risk of heart attack and stroke.

Who statins are indicated for

The ACC/AHA guidelines single out four groups for whom statins are discussed: those with LDL ≥190 mg/dL; those with diabetes aged 40–75; those with established cardiovascular disease; and people aged 40–75 with a 10-year ASCVD risk ≥7.5%. The 7.5% threshold is the point from which the expected benefit usually outweighs the risks.

The decision is always individual: additional risk factors, coronary calcium and patient preferences are taken into account.

Not just cholesterol

Besides lowering LDL, statins have pleiotropic effects: anti-inflammatory, antioxidant, and plaque stabilization. Partly for this reason their benefit is also linked to a reduction in hs-CRP, not only lipids.

Every 1 mmol/L reduction in LDL cuts the risk of major vascular events by about 20%.

Side effects and myths

Most people tolerate statins well. Muscle pain is possible (severe myopathy and rhabdomyolysis are rare), along with a temporary rise in liver enzymes and a small increase in the risk of type 2 diabetes in predisposed people. Real liver damage is rare.

Grapefruit juice and a number of medications raise the concentration of some statins. Stopping abruptly is inadvisable — the risk of events returns.

Reference ranges

Intensity of statin therapy by the expected LDL reduction (ACC/AHA):

High intensityLDL reduction ≥50%
Moderate intensityLDL reduction 30–49%
Low intensityLDL reduction under 30%
Prescription thresholdASCVD risk ≥7.5%
Important: High-intensity regimens include atorvastatin 40–80 mg and rosuvastatin 20–40 mg; the dose choice depends on the level of risk.

Calculate using this marker

Calculators where Statins is used directly:

Frequently asked questions

Will I have to take statins for life?

As a rule, yes: statins control rather than "cure" cholesterol levels, and after stopping, LDL returns to its previous level and the risk of events rises. Discontinuation or a switch is decided with a doctor, not on your own.

Are statins dangerous for the liver?

Serious liver damage is very rare. More often there is an asymptomatic and reversible rise in liver enzymes. Frequent routine ALT monitoring is not needed for most people; the focus is on symptoms and the baseline test.

Related terms

Sources

  1. MedlinePlus — Statins
  2. StatPearls — Statin Medications
info
This content is educational and does not replace consultation with a physician. Reference ranges may vary depending on the laboratory and method — rely on the ranges stated on your own test report.
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